| (210) | Number of the EPO application | 16820497 |
| (220) | Filing date of the EPO application | 2016.12.14 |
| (80) | EPO patent specification publication (B) | EPB nr. 35/2020, 2020.08.26 |
| (110) | EPO patent number | 3390374 |
| (21) | Number of the application | e 2018 1005 |
| (71) | Name(s) of applicant(s), code of the country | MERCK SHARP & DOHME LLC, US; |
| (72) | Name(s) of inventor(s), code of the country | GRESHOCK Thomas J., US;
MULHEARN James, US;
ZHENG Junying, US;
KIM Ronald M., US;
ZHANG Ting, US;
ROECKER Anthony J., US;
WON Walter, US;
NANTERMET Philippe, US;
ANAND Rajan, US;
ZHOU Gang, US;
WANG Deping, US;
GUO Liangqin, US; |
| (73) | Name(s) of owner(s), code of the country | MERCK SHARP & DOHME CORP., US; |
| (54) | Title of the invention | HYDROXYALKYLAMINE- AND HYDROXYCYCLOALKYLAMINE-SUBSTITUTED DIAMINE-ARYLSULFONAMIDE COMPOUNDS WITH SELECTIVE ACTIVITY IN VOLTAGE-GATED SODIUM CHANNELS |
| (13) | Kind-of-document code | A1 |
| (51) | International Patent Classification | C07D 285/08 (2006.01.01); C07D 417/12 (2006.01.01); C07D 277/52 (2006.01.01); A61K 31/4168 (2006.01.01); A61K 31/4178 (2006.01.01); A61K 31/4196 (2006.01.01); A61K 31/551 (2006.01.01); A61P 29/00 (2006.01.01); A61P 11/14 (2006.01.01) |
| (19) | Country | US |
| (41) | Date of publication of the application | 2018.11.30 |
| (30) | Priority | 201562269327 P, 2015.12.18, US; 201662290235 P, 2016.02.02, US; 201662420956 P, 2016.11.11, US |
| (86) | International application | PCT/US2016/066445, 2016.12.14 |
| (87) | International publication | WO 2017/106226, 2017.06.22 |