| (11) | Number of the document | 1507 |
| (21) | Number of the application | 96-0141 |
| (22) | Filing date of the application | 1994.10.07 |
| | Date of filing the request for examination | (pe raspunderea solicitantului) 22.09.1998 |
| (71) | Name(s) of applicant(s), code of the country | AGOURON PHARMACEUTICALS INC., US; |
| (72) | Name(s) of inventor(s), code of the country | DRESSMAN Bruce, A., US; FRITZ James, E., US; HAMMOND Marlys, GB; HORNBACK William, J., US; KALDOR Stephen, W., US; KALISH Vincent, J., US; MUNROE John, E., US; REICH Siegfried, Heinz, US; TATLOCK John Howard, US; SHEPHERD Timothy, A., US; RODRIGUEZ Michael, J., US; JUNGHEIM Louis, N., US; |
| (73) | Name(s) of owner(s), code of the country | AGOURON PHARMACEUTICALS INC., US; |
| (54) | Title of the invention | Inhibitors, pharmaceutical composition on base thereof and process for HIV protease inhibition |
| (13) | Kind-of-document code | |
| (51) | International Patent Classification | A61P 29/00 (2006.01); C07D 217/26 (2006.01); C07D 401/06 (2006.01); C07D 495/04 (2006.01); C07F 9/62 (2006.01); |
| (19) | Country | US |
| (41) | Date of publication of the application | 1998.06.30 |
| (45) | Date of publication of patent granting decision: | 2000.07.31 |
| (47) | Date of issuance of patent | 2001.05.31 |
| (30) | Priority | 08/133,543, 1993.10.07, US; 08/133,696, 1993.10.07, US; 08/190,764, 1994.02.02, US |
| (74) | Patent attorney | SIMANENKOVA Tatiana, Str. Andrei Doga 2/1, MD-2024, Chişinău, Republica Moldova |
| | Substantive examiner(s) | EGOROV Tamara |
| (85) | Date of introducing the national procedure | 1996.03.27 |
| (86) | International application | PCT/US1994/011307, 1994.10.07 |
| (87) | International publication | WO 1995/09843, 1995.04.13 |
| | Expired patents; Date of expiration | 2015.02.28 |
| | Payment for maintenance up to the date | 2014.10.07 |